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Cat. No.: HY-118279

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KSCM-1

KSCM-1 is a selective sigma-1 receptor ligand with a K_i of 27.5 nM. KSCM-1 shows more selective for sigma-1 over sigma-2, and shows no significant affinity at non-sigma receptors.

For research use only. We do not sell to patients.

CAS No.: 1415247-17-4
Formula: C₂₆H₃₂N₂O₄
Molecular Weight:436.54

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

KSCM-1 Chemical Structure

CAS No.: 1415247-17-4

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

KSCM-1 is a selective sigma-1 receptor ligand with a K_i of 27.5 nM. KSCM-1 shows more selective for sigma-1 over sigma-2, and shows no significant affinity at non-sigma receptors^[1].

IC₅₀ & Target^[1]

Sigma 1 Receptor

27.5 nM (Ki)

Sigma 2 Receptor

528 nM (Ki)

All Sigma Receptor Isoforms :

Chemical Information

CAS No. 1415247-17-4
Molecular Weight 436.54
Formula C₂₆H₃₂N₂O₄
SMILES

O=C(N(CCCN1CCCCC1)C2=CC=CC=C2)C3=C(C4=CC(OC)=C(C=C4O3)OC)C
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Karla-Sue C Marriott, et al. Synthesis of N-phenyl-N-(3-(piperidin-1-yl)propyl)benzofuran-2-carboxamides as new selective ligands for sigma receptors. Bioorg Med Chem. 2012 Dec 1;20(23):6856-61. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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KSCM-1

All Sigma Receptor Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

KSCM-1 Related Classifications

HY-118279 Related Classifications