909416-67-7
Chemical Structure
GSK494581A
- CAS. Nr.: 909416-67-7
- Formula:C27H28F2N2O4S
- Molecular Weight:514.58
IUPAC Name: (4-(2-fluoro-4-(1-methoxyethyl)phenyl)piperazin-1-yl)(4'-fluoro-4-(methylsulfonyl)-[1,1'-biphenyl]-2-yl)methanone
InChIKey: JQXZHDOSMUZLML-UHFFFAOYSA-N
SMILES: O=C(N1CCN(C2=CC=C(C(OC)C)C=C2F)CC1)C3=CC(S(=O)(C)=O)=CC=C3C4=CC=C(F)C=C4
Biological Activity: GSK494581A is a specific ligand for human GPR55 (pEC50 of 6.8) and also acts as an inhibitor of glycine transporter subtype 1 (GlyT1). GSK494581A may regulate pain signaling, bone morphogenesis, and vascular endothelial cell formation by binding to GPR55[1].
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GSK494581A | GSK494581A is a specific ligand for human GPR55 (pEC50 of 6.8) and also acts as an inhibitor of glycine transporter subtype 1 (GlyT1). GSK494581A may regulate pain signaling, bone morphogenesis, and vascular endothelial cell formation by binding to GPR55. | |||||||||||||||||||||
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Keywords
