BMS-986034
BMS-986034 is an orally active ingredient (API) that is an agonist of GPR119..
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 1492631-88-5
- Fòrmula: C24H24Cl2N6O4
- Peso molecular:531.39
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
GPR119[1]
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
3 nM
Compound: 4
|
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
|
[PMID: 24900860] |
Chemical Information
-
No. CAS 1492631-88-5
-
Peso molecular 531.39
-
Fòrmula C24H24Cl2N6O4
-
SMILES
O=C1C=C(C(Cl)=CN1C2=NC(C)=C(C=C2)N3C([C@@H](CC3)O)=O)OC4CCN(CC4)C5=NC=C(C=N5)Cl
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)