SB-436811
SB-436811 is a human urotensin-II receptor antagonist with a pKi value of 6.7.
For research use only. We do not sell to patients.
- CAS No.: 346729-66-6
- Formula: C23H29Cl2N3O2
- Molecular Weight:450.40
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | IC50 |
170 nM
Compound: 2a
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Antagonist activity at human recombinant urotensin 2 receptor expressed in HEK293 cells assessed as inhibition of urotensin 2-induced calcium mobilization by FLIPR assay
Antagonist activity at human recombinant urotensin 2 receptor expressed in HEK293 cells assessed as inhibition of urotensin 2-induced calcium mobilization by FLIPR assay
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[PMID: 18573659] |
Chemical Information
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CAS No. 346729-66-6
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Molecular Weight 450.40
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Formula C23H29Cl2N3O2
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SMILES
O=C(C1=CC(Cl)=C(C=C1)Cl)N[C@@H](CC2)CN2CC3=CC=C(C=C3)OCCCN(C)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
SB-436811 Related Classifications
HY-10666 Related Classifications
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