Relzomostat
Relzomostat (Example 18) is a methionyl aminopeptidase 2 (MetAP2) inhibitor. Relzomostat is used for research on obesity and type 2 diabetes.
For research use only. We do not sell to patients.
- CAS No.: 2081078-92-2
- Formula: C24H36F2N2O5
- Molecular Weight:470.55
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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MetAp2 |
MetAP2 is an intracellular Mn2+/Co2+-dependent metalloprotease that catalyzes the cleavage of the N-terminal initiating Met from nascent polypeptides and participates in the regulation of endothelial cell proliferation, lipid metabolism, and insulin sensitivity[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2081078-92-2
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Molecular Weight 470.55
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Formula C24H36F2N2O5
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SMILES
C[C@]1([C@H](O1)C/C=C(C)\C)[C@]2([H])[C@]3(CC[C@H]([C@H]2OC)OC(N4CC5(CN(C5)CC(F)F)C4)=O)CO3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)