CGP52432 (Standard)
CGP52432 (Standard) is the analytical standard of CGP52432 (HY-103531). This product is intended for research and analytical applications. CGP52432 is a GABAB receptor antagonist, with an IC50 of 85 nM.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 139667-74-6
- 分子式: C15H24Cl2NO4P
- 分子量:384.24
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
Product Information
The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
化学情報
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CAS 番号 139667-74-6
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分子量 384.24
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分子式 C15H24Cl2NO4P
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SMILES
O=P(C(OCC)OCC)(CCCNCC1=CC=C(Cl)C(Cl)=C1)O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
[1]. Lanza M, et al. CGP 52432: a novel potent and selective GABAB autoreceptor antagonist in rat cerebral cortex. Eur J Pharmacol. 1993 Jun 24;237(2-3):191-5. [Content Brief]
[2]. Sweeney FF, et al. Activation but not blockade of GABAB receptors during early-life alters anxiety in adulthood in BALB/c mice. Neuropharmacology. 2014 Jun;81:303-10. [Content Brief]
[3]. Kobuchi S, et al. Mechanisms underlying the renoprotective effect of GABA against ischaemia/reperfusion-induced renal injury in rats. Clin Exp Pharmacol Physiol. 2015 Mar;42(3):278-86. [Content Brief]
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)