GPR17 agonist 2
GPR17 agonist 2 (compound 10) is a human GPR17 agonist and selective P2Y receptor non-activator.GPR17 agonist 2 modulates intracellular cAMP levels through functional activation of its target receptor.GPR17 agonist 2 can be used for the research of multiple sclerosis, cerebral ischemia, traumatic brain injury, spinal cord injury.
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- 화학식: C19H32Cl2N9O12P3
- 분자량:742.34
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- 순도&문서
- References
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Help & FAQs
Biological Activity
GPR17 agonist 2 (compound 10) (dose-response curve for EC50 determination) is a potent, full agonist of human GPR17 in HEK293 L9-2 cells, with an EC50 of 62 pM, and shows high selectivity for human GPR17 over human P2Y12, P2Y13, and P2Y14 receptors[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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분자량 742.34
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화학식 C19H32Cl2N9O12P3
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SMILES
O=P(OP(C(Cl)(Cl)P([O-])([O-])=O)([O-])=O)([O-])OC[C@@H]1[C@@H](O)[C@@H](O)[C@H](N2C=NC3=C(N)N=C(C#CC4=CC=CC=C4)N=C32)O1.[NH4+].[NH4+].[NH4+].[NH4+]
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
GPR17 agonist 2 Related Classifications
HY-181738 Related Classifications
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