1. GPCR/G Protein
    Neuronal Signaling
  2. Melanocortin Receptor
  3. MSG606 TFA

MSG606 TFA 

Cat. No.: HY-P1726A
Handling Instructions

MSG606 TFA is a potent human MC1 receptor antagonist (IC50=17 nM). MSG606 TFA also partial agonist at human MC3 and MC5 receptors (EC50 values are 59 and 1300 nM, respectively). MSG606 TFA exhibits binding affinity for A375 melanoma cells in vitro. MSG606 TFA reverses morphine-induced hyperalgesia in female mice, with no effect in male mice.

For research use only. We do not sell to patients.

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MSG606 TFA Chemical Structure

MSG606 TFA Chemical Structure

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Description

MSG606 TFA is a potent human MC1 receptor antagonist (IC50=17 nM). MSG606 TFA also partial agonist at human MC3 and MC5 receptors (EC50 values are 59 and 1300 nM, respectively). MSG606 TFA exhibits binding affinity for A375 melanoma cells in vitro. MSG606 TFA reverses morphine-induced hyperalgesia in female mice, with no effect in male mice.

Molecular Weight

1461.53

Formula

C₆₃H₈₃F₃N₂₀O₁₅S

Sequence

Bua-Gly-His-{d-Phe}-Arg-{d-Trp}-Cys-Asp-Arg-Phe-Gly-NH2 (Carba sulfide bridge:Bua1-Cys7)

Sequence Shortening

{Bua}GH-{d-Phe}-R-{d-Trp}-CDRFG-NH2 (Carba sulfide bridge:Bua1-Cys7)

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

MSG606MSG 606MSG-606Melanocortin ReceptorMC ReceptorInhibitorinhibitorinhibit

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MSG606 TFA
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HY-P1726A
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