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8 Results for "
FAD286
" in MedChemExpress (MCE) Product Catalog:
Products (8)
8 Results for "FAD286" in MCE Product Catalog:
3
3 Cited Publications
Synonyms: CGS 16949A; (Rac)-FAD286 hydrochloride
Target:
Research Areas:
Fadrozole hydrochloride (CGS 16949A) is a potent, selective and nonsteroidal inhibitor of aromatase with an IC50 of 6.4 nM.
3
3 Cited Publications
Synonyms: CGS 16949A free base; (Rac)-FAD286
Target:
Research Areas:
Fadrozole (CGS 16949A free base) is a potent, selective and nonsteroidal inhibitor of aromatase with an IC50 of 6.4 nM.
3
3 Cited Publications
Cat. No.: HY-14247B
CAS No.: 176702-70-8
Synonyms: CGS 16949A hemihydrate; (Rac)-FAD286 hydrochloride hemihydrate
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Research Areas:
Fadrozole hydrochloride hemihydrate is an orally active, potent, selective and nonsteroidal aromatase inhibitor, with an IC50 of 6.4 nM. Fadrozole hydrochloride hemihydrate inhibits the production of estrogen and progesterone, with IC50 values of 0.03 and 120 μM. Fadrozole hydrochloride hemihydrate shows prevention of spontaneous tumours. Fadrozole hydrochloride hemihydrate can be used for the research of estrogen-dependent disease and cancer .
Synonyms: (R)-FADrozole; (R)-CGS 16949A free base; FAD286
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Research Areas:
Dexfadrostat ((R)-Fadrozole) is an orally active and selective aromatase inhibitor, with human aromatase IC50 values of 6.4 nM. Dexfadrostat suppresses estrogen synthesis, reduces circulating estradiol levels and suppresses aldosterone production. Dexfadrostat can be used for the research of breast cancer, primary aldosteronism, and hypertension .
Cat. No.: HY-113986C
CAS No.: 131863-75-7
Synonyms: (R)-FADrozole hydrochloride; (R)-CGS 16949A; FAD286 hydrochloride
Target:
Research Areas:
Dexfadrostat ((R)-Fadrozole) hydrochloride is an orally active and selective aromatase inhibitor, with human aromatase IC50 values of 6.4 nM. Dexfadrostat hydrochloride suppresses estrogen synthesis, reduces circulating estradiol levels and suppresses aldosterone production. Dexfadrostat hydrochloride can be used for the research of breast cancer, primary aldosteronism, and hypertension .
Cat. No.: HY-14247R
CAS No.: 102676-31-3
Synonyms: CGS 16949A (Standard); (Rac)-FAD286 hydrochloride (Standard)
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Research Areas:
Fadrozole (hydrochloride) (Standard) is the analytical standard of Fadrozole (hydrochloride). This product is intended for research and analytical applications. Fadrozole hydrochloride (CGS 16949A) is a potent, selective and nonsteroidal inhibitor of aromatase with an IC50 of 6.4 nM.
Cat. No.: HY-14247AR
CAS No.: 102676-47-1
Synonyms: CGS 16949A free base (Standard); (Rac)-FAD286 (Standard)
Target:
Research Areas:
Fadrozole (Standard) is the analytical standard of Fadrozole. This product is intended for research and analytical applications. Fadrozole (CGS 16949A free base) is a potent, selective and nonsteroidal inhibitor of aromatase with an IC50 of 6.4 nM.
Cat. No.: HY-113986B
CAS No.: 102676-86-8
Synonyms: (S)-FADrozole; (S)-CGS 16949A free base; (S)-FAD286
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Research Areas:
(S)-Dexfadrostat ((S)-Fadrozole) is an aromatase inhibitor with an IC50 of 4.6 nM in human placental microsomes in vitro. (S)-Dexfadrostat can be used in the study of estrogen-dependent breast cancer, gynecomastia, and systemic lupus erythematosus .
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