2 Results for "

1191908-14-1

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "1191908-14-1" in MCE Product Catalog:

Cat. No.: HY-135270
CAS No.: 1191908-14-1
Purity:  98.13%
Target:  

Adrenergic Receptor

Research Areas:  

Endocrinology

ADRA1D receptor antagonist 1 is a potent, selective and orally active α1D adrenoceptor antagonist, with a Ki of 1.6 nM .
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Cat. No.: HY-148252
CAS No.: 1191908-24-3
Target:  

Adrenergic Receptor

Research Areas:  

Endocrinology

ADRA1D receptor antagonist 1 (free base) (compound (R)-9s) is an orally active, potent and selective human α1D-adrenoceptor (α1D-AR) antagonist (Ki=1.6 nM). ADRA1D receptor antagonist 1 (free base) dose-dependently inhibits bladder contraction with an IC30 value of 15 nM. ADRA1D receptor antagonist 1 (free base) can be used in studies of overactive bladder disorders such as urinary urgency, frequency and incontinence.
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