3 Results for "

Anti-inflammatory agent 8

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Anti-inflammatory agent 8" in MCE Product Catalog:

Cat. No.: HY-115920
CAS No.: 1103920-19-9
Target:  

COX

Research Areas:  

Inflammation/Immunology

Anti-inflammatory agent 8 (compound 13) is a tilomisole-based benzimidazothiazole derivative. Anti-inflammatory agent 8 expresses activity on COX-2 enzyme more than COX-1 with an IC50 of 0.09 nM. Anti-inflammatory agent 8 is orally active .
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Cat. No.: HY-151402
CAS No.: 2978694-22-1
Purity:  95.12%
Target:  

Bacterial

Research Areas:  

Infection

Antimicrobial agent-8 (Compound 15) is a potent antimicrobial agent, and shows potent antimicrobial activity with an MIC range of 2-8 μg/mL against Gram-negative and Gram-positive bacteria. Antimicrobial agent-8 shows anti-inflammatory activity against lipopolysaccharide-induced inflammation.
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Cat. No.: HY-152506
Target:  

Amyloid-β

Research Areas:  

Neurological Disease

Antioxidant agent-8 is an orally active inhibitor of 1-42 deposition. Antioxidant agent-8 inhibits fibril aggregation (IC50=11.15 µM) and promotes fibril disaggregation (IC50=6.87 µM). Antioxidant agent-8 also inhibits Cu 2+-induced Aβ1-42 fibril aggregation (IC50=3.69 µM) and promotes Cu 2+-induced Aβ1-42 fibril disaggregation (IC50=3.35 µM). Antioxidant agent-8 has antioxidant activity, anti-inflammatory activity, biosafety, blood-brain barrier permeability and neuroprotective effect .
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