3 Results for "

D81

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "D81" in MCE Product Catalog:

Cat. No.: HY-15780S1
CAS No.: 1427049-19-1
Purity:  96.48%
Synonyms: OPC-34712-d8-1
Brexpiprazole-d8-1 (OPC-34712-d8-1) is the deuterium labeled Brexpiprazole (HY-15780) . Brexpiprazole (OPC-34712), an atypical orally active antipsychotic agent, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM) .
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Cat. No.: HY-W716520
CAS No.: 1308278-69-4
Synonyms: RGH-188-d8
Cariprazine-d8-1 (RGH-188-d8-1) is the deuterium labeled Cariprazine (HY-14763). Cariprazine is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
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Cat. No.: HY-124368
CAS No.: 1491909-40-0
Target:  

SphK

Research Areas:  

Inflammation/Immunology

RB-042 is a SK1 and SK2 inhibitor with IC50 values of 5.3 μM and 5.0 μM, respectively. RB-042 is applicable to the research of inflammatory diseases .
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