Cariprazine-d8
Based on 1 Customer Validation
Cariprazine-d8-1 (RGH-188-d8-1) is the deuterium labeled Cariprazine (HY-14763). Cariprazine is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
For research use only. We do not sell to patients.
- CAS No.: 1308278-69-4
- Formula: C21H24D8Cl2N4O
- Molecular Weight:435.46
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
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Help & FAQs
Biological Activity
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
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CAS No. 1308278-69-4
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Unlabeled Cas 839712-12-8
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Molecular Weight 435.46
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Formula C21H24D8Cl2N4O
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SMILES
ClC1=C(C=CC=C1Cl)N2CCN(CC2)C([2H])(C[C@H]3CC[C@@H](CC3)NC(N(C([2H])([2H])[2H])C([2H])([2H])[2H])=O)[2H]
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Synonyms
RGH-188-d8
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Cariprazine-d8 Related Classifications
HY-W716520 Related Classifications
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