Cariprazine-d8
Based on 1 Customer Validation
Cariprazine-d8-1 (RGH-188-d8-1) is the deuterium labeled Cariprazine (HY-14763). Cariprazine is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 1308278-69-4
- Fòrmula: C21H24D8Cl2N4O
- Peso molecular:435.46
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
Descripciòn
In Vitro
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Aplicación
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
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No. CAS 1308278-69-4
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Unlabeled CAS 839712-12-8
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Peso molecular 435.46
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Fòrmula C21H24D8Cl2N4O
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SMILES
ClC1=C(C=CC=C1Cl)N2CCN(CC2)C([2H])(C[C@H]3CC[C@@H](CC3)NC(N(C([2H])([2H])[2H])C([2H])([2H])[2H])=O)[2H]
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Synonyms
RGH-188-d8
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)