3 Results for "

GAT107

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "GAT107" in MCE Product Catalog:

Cat. No.: HY-117611
CAS No.: 1476807-74-5
Target:  

nAChR

Research Areas:  

Neurological Disease

GAT107 (compound 1b) is a potent α7 nAChR ago-PAMs (positive allosteric modulators) .
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Cat. No.: HY-167922
CAS No.: 1426240-47-2
Target:  

Endogenous Metabolite

Research Areas:  

Neurological Disease

(R,R,S)-GAT107 is a fully agonistic positive modulator of α7 nicotinic receptors with significant biological activity. Its activity is entirely present in its (+)-isomer 1b, while (-)-isomer 1a does not affect its activity when used together. Studies have shown that (R,R,S)-GAT107 is the most potent ago-PAM for α7 nicotinic receptors currently known and has the potential for further in vivo evaluation .
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Cat. No.: HY-167922S
Heptadecanoyl L-carnitine-d3 HCl is the deuterium labeled (R,R,S)-GAT107 (HY-167922). (R,R,S)-GAT107 is a fully agonistic positive modulator of α7 nicotinic receptors with significant biological activity. Its activity is entirely present in its (+)-isomer 1b, while (-)-isomer 1a does not affect its activity when used together. Studies have shown that (R,R,S)-GAT107 is the most potent ago-PAM for α7 nicotinic receptors currently known and has the potential for further in vivo evaluation .
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