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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
4 Results for "
H2-histamine
" in MedChemExpress (MCE) Product Catalog:
Products (4)
4 Results for "H2-histamine" in MCE Product Catalog:
Cat. No.: HY-122148
CAS No.: 83184-14-9
Target:
Research Areas:
DA 4626 is a competitive H2-histamine receptor antagonist. DA 4626 inhibits adenylate cyclase activity with a KB value of 40 nM .
Cat. No.: HY-176060
CAS No.: 1029802-21-8
Research Areas:
Platelet aggregation-IN-3 (Compound 5) is a ligand for H2 histamine receptors, α2(A,C)-adrenergic receptors (α2-AR), and 5-HT2(B,C) serotonin receptors. Platelet aggregation-IN-3 can inhibit platelet aggregation induced by ADP and collagen and can also modulate tumour cell-induced platelet aggregation (TCIPA). Platelet aggregation-IN-3 is promising for research of antiplatelet therapy in cardiovascular diseases and the prevention of cancer-related thrombosis and tumour metastasis .
Cat. No.: HY-101745
CAS No.: 91833-49-7
Synonyms: AHR-11325
Target:
Research Areas:
Rocastine (AHR-11325 ) is an orally active H1-histamine receptor inhibitor that selectively binds to and functionally inhibits H1-histamine receptors. Rocastine protects guinea pigs from the lethal effect induced by Histamine (HY-B1204), prevents histamine-induced collapse, and protects guinea pigs from the falling reaction induced by nebulized antigens. Rocastine can be used in the research of allergic diseases .
Cat. No.: HY-101745B
CAS No.: 91833-50-0
Synonyms: AHR-11325 fumarate
Target:
Research Areas:
Rocastine fumarate (AHR-11325 fumarate) is an orally active H1-histamine receptor inhibitor that selectively binds to and functionally inhibits H1-histamine receptors. Rocastine fumarate protects guinea pigs from the lethal effect induced by Histamine (HY-B1204), prevents histamine-induced collapse, and protects guinea pigs from the falling reaction induced by nebulized antigens. Rocastine fumarate can be used in the research of allergic diseases .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
