91833-50-0
Chemical Structure
Rocastine fumarate
Synonym(s): AHR-11325 fumarate
- CAS No.: 91833-50-0
- Formula:C17H23N3O5S
- Molecular Weight:381.45
IUPAC Name: 2-(2-(dimethylamino)ethyl)-4-methyl-3,4-dihydropyrido[3,2-f][1,4]oxazepine-5(2H)-thione fumarate
InChIKey: LZFCSDIBLCSFAK-WLHGVMLRSA-N
SMILES: OC(/C=C/C(O)=O)=O.S=C1C2=CC=CN=C2OC(CN1C)CCN(C)C
Biological Activity: Rocastine fumarate (AHR-11325 fumarate) is an orally active H1-histamine receptor inhibitor that selectively binds to and functionally inhibits H1-histamine receptors. Rocastine fumarate protects guinea pigs from the lethal effect induced by Histamine (HY-B1204), prevents histamine-induced collapse, and protects guinea pigs from the falling reaction induced by nebulized antigens. Rocastine fumarate can be used in the research of allergic diseases[1].
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Rocastine fumarate | Rocastine fumarate (AHR-11325 fumarate) is an orally active H1-histamine receptor inhibitor that selectively binds to and functionally inhibits H1-histamine receptors. Rocastine fumarate protects guinea pigs from the lethal effect induced by Histamine (HY-B1204), prevents histamine-induced collapse, and protects guinea pigs from the falling reaction induced by nebulized antigens. Rocastine fumarate can be used in the research of allergic diseases. | |||||||||||||||||||||
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