2 Results for "

KOR agonist2

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "KOR agonist2" in MCE Product Catalog:

Cat. No.: HY-159088
CAS No.: 3050912-29-0
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

KOR agonist 2 (Compound 23p) is an agonist for κ opioid receptor (KOR) with Ki of 1.9 nM. KOR agonist 2 exhibits analgesic effect in mouse models with ED50 of 1.30 mg/kg. KOR agonist 2 exhibits high clearance rate (2 mg/kg, i.v.) in mice, high metabolism and clearance in liver microsomes .
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Cat. No.: HY-162552
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

KOR/DOR agonist 2 is a KOR and DOR opioid receptors agonist with Ki values of 0.14 nM, and 0.93 nM, respectively. KOR/DOR agonist 2 shows significant antinociceptive effects. KOR/DOR agonist 2 penetrates the blood-brain barrier .
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