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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
5 Results for "
MSI1436
" in MedChemExpress (MCE) Product Catalog:
Products (5)
5 Results for "MSI1436" in MCE Product Catalog:
Cat. No.: HY-12219
CAS No.: 186139-09-3
Synonyms: Trodusquemine; Aminosterol-1436
Target:
Research Areas:
MSI-1436 is a selective, non-competitive inhibitor of the enzyme protein-tyrosine phosphatase 1B (PTP1B), with an IC50 of appr 1 μM, 200-fold preference over TCPTP (IC50, 224 μM).
8
8 Cited Publications
Synonyms: Trodusquemine lactate; Aminosterol-1436 lactate
Target:
Research Areas:
MSI-1436 lactate is a selective, non-competitive inhibitor of the enzyme protein-tyrosine phosphatase 1B (PTP1B), with an IC50 of 1 μM, 200-fold preference over TCPTP (IC50 of 224 μM).
Target:
Research Areas:
DPM-1001 is a potent, specific, orally active and non-competitive inhibitor of protein-tyrosine phosphatase (PTP1B) with an IC50 of 100 nM. DPM-1001 is an analog of the specific PTP1B inhibitor MSI-1436. DPM-1001 has anti-diabetic property .
Cat. No.: HY-121515A
Purity: 98.48%
Target:
Research Areas:
DPM-1001 trihydrochloride is a potent, specific, orally active and non-competitive inhibitor of protein-tyrosine phosphatase (PTP1B) with an IC50 of 100 nM. DPM-1001 trihydrochloride is an analog of the specific PTP1B inhibitor MSI-1436. DPM-1001 trihydrochloride has anti-diabetic property .
Cat. No.: HY-12219B
CAS No.: 390808-64-7
Target:
Research Areas:
MSI-1701 is an analogue of MSI-1436 which can control weight gain and blood glucose level extracted from patent US 7410959 B1.
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Protocols
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