7 Results for "

Mefloquine

" in MedChemExpress (MCE) Product Catalog:
Products (7)

7 Results for "Mefloquine" in MCE Product Catalog:

4
4 Cited Publications
Cat. No.: HY-17437
CAS No.: 53230-10-7
Synonyms: Mefloquin
Mefloquine (Mefloquin), an orally active and potent quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine is also a K + channel (KvQT1/minK) antagonist with an IC50 of ~1 μM. Mefloquine can be used for malaria, systemic lupus erythematosus and cancer research .
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4
4 Cited Publications
Cat. No.: HY-17437A
CAS No.: 51773-92-3
Synonyms: Mefloquin hydrochloride
Mefloquine hydrochloride (Mefloquin hydrochloride), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine hydrochloride is also a K + channel (KvQT1/minK) antagonist with an IC50 of ~1 μM. Mefloquine hydrochloride can be used for malaria, systemic lupus erythematosus and cancer research .
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Cat. No.: HY-17437R
CAS No.: 53230-10-7
Synonyms: Mefloquin (Standard)
Mefloquine (Standard) is the analytical standard of Mefloquine. This product is intended for research and analytical applications. Mefloquine (Mefloquin), an orally active and potent quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine is also a K+ channel (KvQT1/minK) antagonist with an IC50 of ~1 μM. Mefloquine can be used for malaria, systemic lupus erythematosus and cancer research .
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Cat. No.: HY-17437AR
CAS No.: 51773-92-3
Synonyms: Mefloquin hydrochloride (Standard)
Mefloquine (hydrochloride) (Standard) is the analytical standard of Mefloquine (hydrochloride). This product is intended for research and analytical applications. Mefloquine hydrochloride (Mefloquin hydrochloride), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine hydrochloride is also a K+ channel (KvQT1/minK) antagonist with an IC50 of ~1 μM. Mefloquine hydrochloride can be used for malaria, systemic lupus erythematosus and cancer research .
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Cat. No.: HY-W324493
CAS No.: 35853-50-0
Synonyms: Ro 21-5104
Target:  

Drug Metabolite

Research Areas:  

Infection

Carboxymefloquine is a metabolite of Mefloquine (HY-17437) (an antimalarial agent). Carboxymefloquine can be used in malaria research .
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Cat. No.: HY-132651S
CAS No.: 1246819-32-8
Dehydro Mefloquine-d5 is the deuterium labeled Dehydro Mefloquine .
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Cat. No.: HY-17437C
CAS No.: 49752-90-1
Synonyms: (Rac)-Mefloquin
Target:  

NF-κB IKK Apoptosis

Research Areas:  

Cancer

(Rac)-Mefloquine ((Rac)-Mefloquin) is an orally active NF-κB inhibitor. (Rac)-Mefloquine inhibits the NF-κB and IKK signaling pathways, suppresses NF-κB-Luc luciferase activity, blocks the activation of p65 and IκBα, and reduces the expression of downstream target genes of NF-κB. (Rac)-Mefloquine activates apoptosis-related factors and induces apoptosis in tumor cells. (Rac)-Mefloquine functions as a tumor cell inhibitor. (Rac)-Mefloquine can be used for the research of colorectal cancer .
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