3 Results for "

R 43512

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "R 43512" in MCE Product Catalog:

9
9 Cited Publications
Cat. No.: HY-12532
CAS No.: 68844-77-9
Purity:  99.77%
Synonyms: R 43512
Astemizole (R 43512), a second-generation antihistamine agent to diminish allergic symptoms with a long duration of action, is a histamine H1-receptor antagonist, with an IC50 of 4 nM. Astemizole also shows potent hERG K + channel blocking activity with an IC50 of 0.9 nM. Astemizole has antipruritic effects .
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Cat. No.: HY-12532R
CAS No.: 68844-77-9
Synonyms: R 43512 (Standard)
Astemizole (Standard) is the analytical standard of Astemizole. This product is intended for research and analytical applications. Astemizole (R 43512), a second-generation antihistamine agent to diminish allergic symptoms with a long duration of action, is a histamine H1-receptor antagonist, with an IC50 of 4 nM. Astemizole also shows potent hERG K + channel blocking activity with an IC50 of 0.9 nM. Astemizole has antipruritic effects .
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Cat. No.: HY-12532S
CAS No.: 1189961-39-4
Astemizole-d3 is the deuterium labeled Astemizole. Astemizole (R 43512), a second-generation antihistamine drug to diminish allergic symptoms with a long duration of action, is a histamine H1-receptor antagonist, with an IC50 of 4 nM. Astemizole also shows potent hERG K+ channel blocking activity with an IC50 of 0.9 nM. Astemizole has antipruritic effects .
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