3 Results for "

RG3487

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "RG3487" in MCE Product Catalog:

Cat. No.: HY-108057A
CAS No.: 677305-02-1
Purity:  99.66%
Synonyms: RG3487 hydrochloride
Target:  

nAChR 5-HT Receptor

Research Areas:  

Neurological Disease

Facinicline hydrochloride (RG3487 hydrochloride) is an orally active nicotinic α7 receptor partial agonist, with a Ki of 6 nM for α7 human nAChR. Facinicline hydrochloride (RG3487 hydrochloride) improves cognition and sensorimotor gating in rodents. Facinicline hydrochloride (RG3487 hydrochloride) shows high affinity (antagonist) to 5-HT3Rs with a Ki value of 1.2 nM .
loading...
    loading...
Cat. No.: HY-108057
CAS No.: 677306-35-3
Synonyms: RG3487 free base
Target:  

nAChR 5-HT Receptor

Research Areas:  

Neurological Disease

Facinicline (RG3487) is an orally active nicotinic α7 receptor partial agonist, with a Ki of 6 nM for α7 human nAChR. Facinicline improves cognition and sensorimotor gating in rodents. Facinicline hydrochloride shows high affinity (antagonist) to 5-HT3Rs with a Ki value of 1.2 nM .
loading...
    loading...
Cat. No.: HY-108057AR
CAS No.: 677305-02-1
Synonyms: RG3487 hydrochloride (Standard)
Facinicline hydrochloride (Standard) is the analytical standard of Facinicline (hydrochloride) (HY-108057A). This product is intended for research and analytical applications. Facinicline hydrochloride (RG3487 hydrochloride) is an orally active nicotinic α7 receptor partial agonist, with a Ki of 6 nM for α7 human nAChR. Facinicline hydrochloride (RG3487 hydrochloride) improves cognition and sensorimotor gating in rodents. Facinicline hydrochloride (RG3487 hydrochloride) shows high affinity (antagonist) to 5-HT3Rs with a Ki value of 1.2 nM .
loading...
    loading...