2 Results for "

hM2R

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "hM2R" in MCE Product Catalog:

8
8 Cited Publications
Cat. No.: HY-17585
CAS No.: 76-90-4
Target:  

mAChR GPR109A

Research Areas:  

Others Inflammation/Immunology

Mepenzolate bromide is an orally administered muscarinic receptor antagonist with Kis of 0.68 and 2.6 nM for hM2R and hM3R, respectively. Mepenzolate bromide can be used to suppress the gastrointestinal hypermotility associated with irritable bowel syndrome .Mepenzolate bromide is a GPR109A inhibitor [2].
loading...
    loading...
Cat. No.: HY-170444
Research Areas:  

Neurological Disease

ADS1017 is the antagonist for histamine receptor and muscarinic receptor, that exhibits good affinities to hH3R, hH4R, hM2R and hM4R with pKi of 6.8, 5.5, 7.4 and 7.2. ADS1017 exhibits analgesic and anti-allodynic efficacy in mice Capsaicin (HY-10448)-or Oxaliplatin (HY-17371)-induced pain models .
loading...
    loading...