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Cat. No.: HY-19924

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GSK-1440115

GSK-1440115 is an antagonist of the Urotensin II Receptor with an IC₅₀ value of 82.3 nM.

For research use only. We do not sell to patients.

CAS No.: 1003878-16-7
Formula: C₃₀H₂₉Cl₂N₃O₆
Molecular Weight:598.47

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

GSK-1440115 Chemical Structure

CAS No.: 1003878-16-7

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

GSK-1440115 is an antagonist of the Urotensin II Receptor with an IC₅₀ value of 82.3 nM^[1].

Chemical Information

CAS No. 1003878-16-7
Molecular Weight 598.47
Formula C₃₀H₂₉Cl₂N₃O₆
SMILES

O=C(C1=CC=C(C2=CC=C([C@@H](N(C(CN3C(COC4=CC(Cl)=C(Cl)C=C34)=O)=O)C)CN5CCOCC5)C=C2)C=C1)O
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Tae-Ho Kim, et al. A Novel Urotensin II Receptor Antagonist, KR-36996 Inhibits Smooth Muscle Proliferation through ERK/ROS Pathway. Biomol Ther (Seoul). 2017 May 1;25(3):308-314. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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