1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. FGFR
  4. FGFR4 Inhibitors

FGFR4 Inhibitors

FGFR

FGFR1

FGFR2

FGFR3

FGFR4

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform FGFR4 together.

Please try each isoform separately.

FGFR4 Specific Inhibitors
Product Name FGFR4 FGFR1 FGFR2 FGFR3 FGFR4 Selectivity Purity
Roblitinib
FGFR4, IC50: 1.9 nM
      Selective Inhibitor 98.08%
FGFR4-IN-1
FGFR4, IC50: 0.7 nM
      Selective Inhibitor 99.93%
Infigratinib
FGFR4, IC50: 60 nM
FGFR1, IC50: 0.9 nM
FGFR2, IC50: 1.4 nM
FGFR3, IC50: 1 nM
Pan Inhibitor 99.16%
AZD4547
FGFR4, IC50: 165 nM
FGFR1, IC50: 0.2 nM
FGFR2, IC50: 2.5 nM
FGFR3, IC50: 1.8 nM
Pan Inhibitor 99.80%
LY2874455
FGFR4, IC50: 6 nM
FGFR1, IC50: 2.8 nM
FGFR2, IC50: 2.6 nM
FGFR3, IC50: 6.4 nM
Pan Inhibitor 98.02%
PRN1371
FGFR4, IC50: 19.3 nM
FGFR1, IC50: 0.6 nM
FGFR2, IC50: 1.3 nM
FGFR3, IC50: 4.1 nM
Pan Inhibitor 99.24%
CH5183284
FGFR4, IC50: 290 nM
FGFR1, IC50: 9.3 nM
FGFR2, IC50: 7.6 nM
FGFR3, IC50: 22 nM
Pan Inhibitor 99.73%
FIIN-2
FGFR4, IC50: 45 nM
FGFR1, IC50: 3.1 nM
FGFR2, IC50: 4.3 nM
FGFR3, IC50: 27 nM
Pan Inhibitor 99.95%
Infigratinib phosphate
FGFR4, IC50: 60 nM
FGFR1, IC50: 0.9 nM
FGFR2, IC50: 1.4 nM
FGFR3, IC50: 1 nM
Pan Inhibitor 97.74%
FIIN-3
FGFR4, IC50: 35.3 nM
FGFR1, IC50: 13.1 nM
FGFR2, IC50: 21 nM
FGFR3, IC50: 31.4 nM
Pan Inhibitor 98.24%
ODM-203
FGFR4, IC50: 35 nM
FGFR1, IC50: 11 nM
FGFR2, IC50: 16 nM
FGFR3, IC50: 6 nM
Pan Inhibitor
ASP5878
FGFR4, IC50: 3.5 nM
FGFR1, IC50: 0.47 nM
FGFR2, IC50: 0.6 nM
FGFR3, IC50: 0.74 nM
Pan Inhibitor 99.71%
Rogaratinib
FGFR4
FGFR1
FGFR2
FGFR3
default Inhibitor 99.38%
Fisogatinib
FGFR4
      default Inhibitor 99.84%