162408-66-4
162408-66-4
Chemical Structure
GR 103691
- CAS No.: 162408-66-4
- Formula:C30H35N3O3
- Molecular Weight:485.62
IUPAC Name: 4'-acetyl-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-[1,1'-biphenyl]-4-carboxamide
InChIKey: JARNORYOPMINDY-UHFFFAOYSA-N
SMILES: O=C(C1=CC=C(C2=CC=C(C(C)=O)C=C2)C=C1)NCCCCN3CCN(C4=CC=CC=C4OC)CC3
Biological Activity: GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
GR 103691 | 99.91% | GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
GR 103691 (Standard) | ≥98% | GR 103691 (Standard) is the analytical standard of GR 103691 (HY-101382). This product is intended for research and analytical applications. GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
Structural Analogs
-
Similarity Score 0.77
HY-116820OS-3-106 -
Similarity Score 0.75
HY-106660BP 897 hydrochloride -
Similarity Score 0.75
HY-114085BP 897 -
Similarity Score 0.67
HY-115968Dopamine D3 receptor ligand-4 -
Similarity Score 0.65
HY-119277CJB-090 dihydrochloride -
Similarity Score 0.65
HY-138809FAUC 346 -
Similarity Score 0.64
HY-180815α1A/1D-Adrenoceptor antagonist-1 -
Similarity Score 0.63
HY-117699RFluanisone (Standard) -
Similarity Score 0.63
HY-146202PDE4B/7A-IN-2 -
Explore the MedChemAI to find more analogs
