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Referencia número: HY-N12399

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Aplithianines A

Aplithianines A is a potent inhibitor against J-PKA_cα with an IC₅₀ of 1 μM , and inhibits wild-type PKA with an IC₅₀ of 84 nM. Aplithianines A inhibits J-PKAcα catalytic activity by competitively binding to the ATP pocket.

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No. CAS: 3027425-38-0
Fòrmula: C₁₃H₁₃N₇S
Peso molecular:299.35

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (269 KB)

Aplithianines A Chemical Structure

No. CAS: 3027425-38-0

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Descripciòn

IC₅₀ & Target

1 μM (J-PKAcα)^[1]

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Chemical Information

No. CAS 3027425-38-0
Peso molecular 299.35
Fòrmula C₁₃H₁₃N₇S
SMILES

CN1C=NC=C1C(SCC2)=CN2C3=NC=NC4=C3N=CN4
Structure Classification
- Alkaloids
- Other Alkaloids
Initial Source
- Microorganisms
Aplidium sp.
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (269 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Du L, et al. Discovery and Synthesis of a Naturally Derived Protein Kinase Inhibitor that Selectively Inhibits Distinct Classes of Serine/Threonine Kinases. J Nat Prod. 2023;86(10):2283-2293. IF: 5.1 Q1 B2 [Content Brief]

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Aplithianines A

Ver todos los productos específicos de isoformas PKA

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Aplithianines A Related Classifications

HY-N12399 Related Classifications