DPP-4-IN-3
DPP-4-IN-3 (Compound 5a) is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 of 0.75 nM. DPP-4-IN-3 shows excellent antioxidant and insulinotropic activity.
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- No. CAS: 2402735-14-0
- Fòrmula: C19H22N6O2
- Peso molecular:366.42
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
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DPP-4 |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| INS1(832/13) | IC50 |
0.0028 μM
Compound: 5a
|
Antidiabetic activity in glucose-treated rat INS1(832/13) cells assessed as increase in insulin release in presence of 3 mM glucose measured after 2 hrs by radioimmunoassay
Antidiabetic activity in glucose-treated rat INS1(832/13) cells assessed as increase in insulin release in presence of 3 mM glucose measured after 2 hrs by radioimmunoassay
|
[PMID: 31812034] |
Chemical Information
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No. CAS 2402735-14-0
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Peso molecular 366.42
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Fòrmula C19H22N6O2
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SMILES
CCOC(N1CCN(CC1)C2=NN3C(C=C2)=NN=C3C4=CC=CC(C)=C4)=O
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)