LSD1-IN-2
LSD1-IN-2 is a LSD1 inhibitor with an IC50 of 0.5 μM. LSD1-IN-2 increases the levels of monomethylated and dimethylated histone H3 lysine 4 (H3K4me1/2) in cells. LSD1-IN-2 reactivates epigenetically silenced tumor suppressor genes. LSD1-IN-2 can be used in the research of colon cancer.
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- No. CAS: 927019-63-4
- Fòrmula: C15H36N8
- Peso molecular:328.51
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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LSD1 0.5 μM (IC50) |
LSD1-IN-2 (Compound 39) potently inhibits LSD1 with an IC50 of 0.5 μM[1].
LSD1-IN-2 (0.5-10 μM) induces dose-dependent increases in H3K4me1/2 levels and tumor suppressor gene re-expression in HCT-116 colon cancer cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 927019-63-4
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Peso molecular 328.51
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Fòrmula C15H36N8
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SMILES
N(=C(NC)NC)CCCNCCCNCCCN=C(NC)NC
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LSD1-IN-2 Related Classifications
HY-124961 Related Classifications
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