Zolertine
Zolertine is an α-adrenergic receptor antagonist, with a pKi of 6.35 for rabbit α1A-adrenergic receptor and a pKi of 6.81 for rat α1B-adrenergic receptor. Zolertine competitively blocks α1D-adrenergic receptor-mediated vasoconstriction and α1A-adrenergic receptor-mediated vasoconstriction in arteries. Zolertine can be used in the research of hypertension.
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- No. CAS: 4004-94-8
- Fòrmula: C13H18N6
- Peso molecular:258.32
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Ver todos los productos específicos de isoformas Adrenergic Receptor
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Actividad biológica
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α1A-adrenergic receptor 6.35 (pKi) |
α1B-adrenergic receptor 6.81 (pKi) |
Zolertine (30 min) competes for the α1-adrenergic receptor binding sites on rat liver (α1B) and rabbit liver (α1A) cell membranes, with pKi values of 6.81 and 6.35, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 4004-94-8
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Peso molecular 258.32
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Fòrmula C13H18N6
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SMILES
C1(CCN2CCN(CC2)C3=CC=CC=C3)=NN=NN1
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Zolertine Related Classifications
HY-183177 Related Classifications
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