AMYR/CTR agonist 1
AMYR/CTR agonist 1 is an amylin receptor (AMYR) and calcitonin receptor (CTR) agonist with an amylin receptor cAMP stimulation EC50 of 0.0995 nM and a calcitonin receptor cAMP stimulation EC50 of 0.00616 nM. AMYR/CTR agonist 1 can be used for the research of non-alcoholic fatty liver disease, non-alcoholic steatohepatitis, insulin dependent diabetes, non-insulin dependent diabetes, impaired glucose tolerance, obesity, syndrome x.
For research use only. We do not sell to patients.
- CAS No.: 3097592-82-7
- Formula: C39H31F3N6O4S
- Molecular Weight:736.76
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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AMYR 99.5 pM (EC50) |
CTR 6.16 pM (EC50) |
AMYR/CTR agonist 1 (compound 195) exhibits agonist activity at both the amylin receptor (cAMP) and the calcitonin receptor (cAMP), with EC50 values of 99.5 pM and 6.16 pM, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3097592-82-7
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Molecular Weight 736.76
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Formula C39H31F3N6O4S
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SMILES
COC1=C(C(F)=CC2=C1CC[C@H]2NC3=NC(C)=CC4=C3SC(C5=C6C(N7CC8CC7(C6=NC(CCC9=CC=C(C=C9)F)=C5C%10=NNC(O%10)=O)C8)=O)=C4)F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
AMYR/CTR agonist 1 Related Classifications
HY-186104 Related Classifications
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