KSL 128114
Based on 1 publication(s) in Google Scholar
KSL 128114, a peptide inhibitor of syntenin, binds the PDZ1 domain of syntenin with nanomolar affinity. KSL 128114 is resistant toward degradation in human plasma and mouse hepatic microsomes and displays a global PDZ domain selectivity for syntenin.
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- CAS 番号: 2757292-12-7
- 分子式: C96H165N39O21
- 分子量:2201.59
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
MedChemExpress（MCE）の使用を引用している文献 KSL 128114
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生物活性
KSL-128114 (~20 μM) shows an inhibitory effect on primary GBM cell viability and significantly extends survival time in a patient-derived xenograft mouse model[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 2757292-12-7
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分子量 2201.59
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分子式 C96H165N39O21
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配列
Ac-{d-Arg}-Arg-{d-Arg}-Gly-{d-Arg}-Lys-{d-Lys}-Arg-{d-Arg}-Ser-His-Trp-{Tle}-{Chg}-Asp-Ile
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シーケンスの短縮
Ac-{d-Arg}-R-{d-Arg}-G-{d-Arg}-K-{d-Lys}-R-{d-Arg}-SHW-{Tle}-{Chg}-DI
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (1)
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Journal Impact Factor
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Most Recent
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Eur J Med Chem
Design, synthesis, and biological evaluation of novel and highly potent peptides targeting syntenin. [Abstract]2025 May 5:289:117446. PMID: 40020425
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
KSL 128114 関連分類
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