RSK2-IN-2
RSK2-IN-2 (Compound 25) is a reversible covalent inhibitor of the RPS6KA3 (RSK2) kinase. RSK2-IN-2 is also described to inhibit MSK1, MSK2 and RSK3.
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- CAS 番号: 1637749-78-0
- 分子式: C16H11N5O
- 分子量:289.29
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
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RSK2 |
RSK3 |
MSK1 |
MSK2 |
RSK2-IN-2 (Compound 25) shows strong activity with ERK2-MSK1 cascade pIC50 of 9.6[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 1637749-78-0
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分子量 289.29
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分子式 C16H11N5O
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SMILES
O=C(N)/C(C#N)=C/C1=CC=CC(C2=C3C(NC=C3)=NC=N2)=C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)