1. Membrane Transporter/Ion Channel
  2. P-glycoprotein
  3. Laniquidar

Laniquidar (Synonyms: R101933)

Cat. No.: HY-132189
Handling Instructions

Laniquidar (R101933) is a noncompetitive, third generation P-glycoprotein (P-gp) inhibitor with an IC50 of 0.51 μM. Laniquidar can be used for modulating multidrug resistance transporters. Laniquidar can also be used for studying acute myeloid leukemia (AML) and myelodysplastic syndrome (MDS). Laniquidar has limited oral bioavailability.

For research use only. We do not sell to patients.

Laniquidar Chemical Structure

Laniquidar Chemical Structure

CAS No. : 197509-46-9

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Description

Laniquidar (R101933) is a noncompetitive, third generation P-glycoprotein (P-gp) inhibitor with an IC50 of 0.51 μM. Laniquidar can be used for modulating multidrug resistance transporters[1]. Laniquidar can also be used for studying acute myeloid leukemia (AML) and myelodysplastic syndrome (MDS)[2]. Laniquidar has limited oral bioavailability[3].

IC50 & Target

IC50: 0.51 μM (P-glycoprotein)[1]

Molecular Weight

584.71

Formula

C37H36N4O3

CAS No.
SMILES

O=C(C1=CN=C2/C(C3=C(CCN21)C=CC=C3)=C4CCN(CC\4)CCC5=CC=C(C=C5)OCC6=NC7=C(C=C6)C=CC=C7)OC

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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