197509-46-9
Chemical Structure
Laniquidar
- CAS No.: 197509-46-9
- Formula:C37H36N4O3
- Molecular Weight:584.71
IUPAC Name: methyl 11-(1-(4-(quinolin-2-ylmethoxy)phenethyl)piperidin-4-ylidene)-6,11-dihydro-5H-benzo[d]imidazo[1,2-a]azepine-3-carboxylate
InChIKey: TULGGJGJQXESOO-UHFFFAOYSA-N
SMILES: O=C(C1=CN=C2/C(C3=C(CCN21)C=CC=C3)=C4CCN(CC\4)CCC5=CC=C(C=C5)OCC6=NC7=C(C=C6)C=CC=C7)OC
Biological Activity: Laniquidar is a non-competitive P-gp inhibitor with an IC50 of 0.51 μM. Laniquidar binds to the P-gp transporter with high affinity and exhibits low activity as a substrate. Laniquidar is applicable to epilepsy-related research[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Laniquidar | 98.86% | Laniquidar is a non-competitive P-gp inhibitor with an IC50 of 0.51 μM. Laniquidar binds to the P-gp transporter with high affinity and exhibits low activity as a substrate. Laniquidar is applicable to epilepsy-related research. | ||||||||||||||||||||
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Keywords