2 Results for "

Altinicline

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Altinicline" in MCE Product Catalog:

Cat. No.: HY-107681
CAS No.: 192231-16-6
Synonyms: SIB-1508Y
Target:  

nAChR

Research Areas:  

Neurological Disease

Altinicline (maleate) is an orally active and selective nAChR agonist. Altinicline (maleate) has the potential to study parkinsonism . Altinicline (maleate) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
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Cat. No.: HY-14318
CAS No.: 179120-92-4
Synonyms: SIB-1508Y free base
Target:  

nAChR

Research Areas:  

Neurological Disease

Altinicline (SIB-1508Y free base) is a selective α4β2 nicotinic acetylcholine receptor (nAChR) agonist, with no activity against α7 or α1β1γδ nAChRs and only extremely low activity against α3β4 nAChRs. Altinicline reverses escape deficits and increases avoidance responses. Altinicline is applicable to research related to depression .
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