4 Results for "

Benzomalvin A

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "Benzomalvin A" in MCE Product Catalog:

Cat. No.: HY-118463
CAS No.: 157047-96-6
Synonyms: (-)-Benzomalvin A
Benzomalvin A is a potent antagonist of neurokinin receptor isolated from Penicillium sp. Benzomalvin A shows inhibitory activity against substance P with Ki values of 12, 42 and 43 μM at the guinea pig, rat and human neurokinin NK1 receptors, respectively .
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Cat. No.: HY-114673
CAS No.: 157047-97-7
Benzomalvin B is the less active analogs of Benzomalvin A. Benzomalvin B is weakly active against substance P .
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Cat. No.: HY-176099
Target:  

Drug Isomer

Research Areas:  

Others

Epibenzomalvin E is an isomer of Benzmalvin E. Benzomalvin E is an indoleamine 2,3-dioxygenase inhibitor .
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Cat. No.: HY-116620
CAS No.: 157047-98-8
Benzomalvin C is a weak antagonist of the neurokinin-1 (NK1) receptor inhibiting binding of substance P by 46% when used at 100 μg/mL in vitro. It is also a weak inhibitor of indolamine 2,3-dioxygenase (IDO) with an IC50 value of 130 μM for recombinant IDO. It is isolated from Penicillium and contains an epoxide group at C-19 and C-20, which is not present in benzomalvins A, B, or E.
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