7 Results for "

Flupenthixol

" in MedChemExpress (MCE) Product Catalog:
Products (7)

7 Results for "Flupenthixol" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-15856B
CAS No.: 2413-38-9
Purity:  98.52%
Synonyms: Flupenthixol dihydrochloride
Research Areas:  

Neurological Disease Cancer

Flupentixol is an orally active D1/D2 dopamine receptor antagonist and new PI3K inhibitor (PI3Kα IC50=127 nM). Flupentixol shows anti-proliferative activity to cancer cells and induces apoptosis. Flupentixol can also be used in schizophrenia, anxiolytic and depressive research .
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Cat. No.: HY-15856A
CAS No.: 2709-56-0
Synonyms: Flupenthixol
Research Areas:  

Neurological Disease

Flupentixol is an orally active D1/D2 dopamine receptor antagonist and new PI3K inhibitor (PI3Kα IC50=127 nM). Flupentixol shows anti-proliferative activity to cancer cells and induces apoptosis. Flupentixol can also be used in schizophrenia, anxiolytic and depressive research .
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Cat. No.: HY-15856
CAS No.: 51529-01-2
Synonyms: cis-(Z)-Flupenthixol dihydrochloride
Research Areas:  

Neurological Disease

cis-(Z)-Flupentixol dihydrochloride is a potent and selective DA D1/D2 receptor antagonist, with Ki values of 0.38 nM and 7 nM for D2 receptor and 5-HT2A, respectively .
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Cat. No.: HY-105657A
CAS No.: 69079-98-7
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

(Z)-Flupenthixol decanoate is the cis form of Flupenthixol decanoate. (Z)-Flupenthixol decanoate is a potent dopamine D1/D2 receptor antagonist. (Z)-Flupenthixol decanoate shows antipsychotic effect .
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Cat. No.: HY-15856BR
CAS No.: 2413-38-9
Synonyms: Flupenthixol dihydrochloride (Standard)
Flupentixol (dihydrochloride) (Standard) is the analytical standard of Flupentixol (dihydrochloride). This product is intended for research and analytical applications. Flupentixol is an orally active D1/D2 dopamine receptor antagonist and new PI3K inhibitor (PI3Kα IC50=127 nM). Flupentixol shows anti-proliferative activity to cancer cells and induces apoptosis. Flupentixol can also be used in schizophrenia, anxiolytic and depressive research .
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Cat. No.: HY-105657
CAS No.: 30909-51-4
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

Flupenthixol decanoate is a dopamine D2 receptor antagonist with antipsychotic effects. Flupenthixol decanoate can be used for schizophrenia and depression research .
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Cat. No.: HY-184837
CAS No.: 53772-82-0
Target:  

Dopamine Receptor

Research Areas:  

Neurological Disease

cis-Flupenthixol is an orally active dopamine receptor antagonist, with a Ki value of 1.4 nM for the Dopamine D-1 receptor and 0.74 nM for the Dopamine D-2 receptor. cis-Flupenthixol blocks dopamine receptors in the medial preoptic area and striatum, impairs male mating behavior, and reduces the concentrations of striatal dopamine metabolites. cis-Flupenthixol alters striatal acetylcholine concentrations in a time-dependent manner and enhances Apomorphine (HY-12723)-induced stereotyped behaviors. cis-Flupenthixol inhibits exploratory locomotor activity and triggers a compensatory increase in dopamine turnover in the striatum and limbic regions. cis-Flupenthixol can be used in studies related to tardive dyskinesia .
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