11 Results for "

Lupeol

" in MedChemExpress (MCE) Product Catalog:
Products (11)

11 Results for "Lupeol" in MCE Product Catalog:

6
6 Cited Publications
Referencia número: HY-N0790
No. CAS: 545-47-1
Synonyms: Clerodol; Monogynol B; Fagarasterol
Lupeol (Clerodol; Monogynol B; Fagarasterol) is an active pentacyclic triterpenoid, has anti-oxidant, anti-mutagenic, anti-tumor and anti-inflammatory activity. Lupeol is a potent androgen receptor (AR) inhibitor and can be used for cancer research, especially prostate cancer of androgen-dependent phenotype (ADPC) and castration resistant phenotype (CRPC) .
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1
1 Cited Publications
Referencia número: HY-126114
No. CAS: 1617-68-1
Pureza:  ≥98.0%
Lupeol acetate is a derivative of Lupeol. Lupeol acetate is an anti-inflammatory, antibacterial, anti-trypanosomic and anticancer agent with oral activity. Lupeol acetate significantly improves the symptoms of rheumatoid arthritis by down-regulating the expression of inflammatory cytokines and osteoclast production. Lupeol acetate inhibits spermatogenesis in male rats and eventually led to infertility .
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Referencia número: HY-N3356
No. CAS: 32214-80-5
Lupeol palmitate is a natural compound with antiulcer activities. Lupeol palmitate has a gastroprotective action .
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Referencia número: HY-N0790R
No. CAS: 545-47-1
Synonyms: Clerodol (Standard); Monogynol B (Standard); Fagarasterol (Standard)
Lupeol (Standard) is the analytical standard of Lupeol. This product is intended for research and analytical applications. Lupeol (Clerodol; Monogynol B; Fagarasterol) is an active pentacyclic?triterpenoid, has anti-oxidant, anti-mutagenic, anti-tumor and anti-inflammatory activity. Lupeol is a potent?androgen receptor (AR)?inhibitor and can be used for cancer research, especially prostate cancer of androgen-dependent phenotype (ADPC) and castration resistant phenotype (CRPC) .
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Referencia número: HY-126114R
No. CAS: 1617-68-1
Lupeol acetate (Standard) is the analytical standard of Lupeol acetate. This product is intended for research and analytical applications. Lupeol acetate is a derivative of Lupeol. Lupeol acetate is an anti-inflammatory, antibacterial, anti-trypanosomic and anticancer agent with oral activity. Lupeol acetate significantly improves the symptoms of rheumatoid arthritis by down-regulating the expression of inflammatory cytokines and osteoclast production. Lupeol acetate inhibits spermatogenesis in male rats and eventually led to infertility .
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Referencia número: HY-W744741
Lupeol-d3 is the deuterium labeled Lupeol (HY-N0790). Lupeol is an active pentacyclic triterpenoid, has anti-oxidant, anti-mutagenic, anti-tumor and anti-inflammatory activity. Lupeol is a potent?androgen receptor?(AR)?inhibitor and can be used for?cancer?research, especially prostate?cancer?of androgen-dependent phenotype (ADPC) and castration resistant phenotype (CRPC) .
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Referencia número: HY-N3358
No. CAS: 108885-61-6
Lupeol β-hydroxyoctadecanoate is a Triterpenoids product that can be isolated from the roots of Biondia hemsleyana. .
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Referencia número: HY-N1824
No. CAS: 29028-10-2
Synonyms: 1β-Hydroxy-Lupeol
3-Epiglochidiol (1β-Hydroxy-lupeol) is a Alkaloids product that can be isolated from the barks of Pandanus amaryllifolius .
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Referencia número: HY-163485
No. CAS: 3036567-30-0
Target:  

Androgen Receptor

Áreas de investigación:  

Endocrinology

AR antagonist 8 (compound 16), an unnatural entestrane, is a potent Lupeol-inspired androgen receptor (AR) antagonist with an IC50 of 0.76 μM .
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Referencia número: HY-E71273
Áreas de investigación:  

Others

β-Amyrin synthase (EC 5.4.99.39) catalyses the synthesis of α-amyrin (EC 5.4.99.40) or lupeol (EC 5.4.99.41) .
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Referencia número: HY-E71272
Áreas de investigación:  

Others

β-Amyrin 28-monooxygenase (EC 1.14.13.201), found in plants, is involved in the biosynthesis of oleanane-type triterpenoids, such as ginsenoside Ro. The enzyme from Medicago trunculata (CYP716A12) can also convert α-amyrin and lupeol to ursolic acid and betulinic acid, respectively.
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