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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
5 Results for "
human GPR52
" in MedChemExpress (MCE) Product Catalog:
Products (5)
5 Results for "human GPR52" in MCE Product Catalog:
Target:
Research Areas:
NXE0041178 is an orally active and BBB-penetrant full GPR52 agonist, with a pEC50 of 7.5 for human GPR52 and an EC50 of 27.5 nM (pEC50 = 7.55) for rat GPR52. NXE0041178 shows no significant inhibition on hERG, hNaV1.5 and cytochrome P450 isoforms. NXE0041178 can reduce d-amphetamine-induced hyperactivity in rats. NXE0041178 can be used for research of Neurological disease .
Cat. No.: HY-RS05718
Target:
Research Areas:
GPR52 Human Pre-designed siRNA Set A contains three designed siRNAs for GPR52 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-163671
CAS No.: 2767348-36-5
Research Areas:
PW0729 is a selective GPR52 agonist. PW0729 activates G protein/cAMP signaling pathway, with bias toward this pathway over β-arrestin recruitment, and induces GPR52 desensitization. PW0729 can be used for the research of neuropsychiatric and neurological diseases .
Cat. No.: HY-P703263
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: GPR52; G-Protein Coupled Receptor 52; G Protein-Coupled Receptor 52; Probable G-Protein Coupled Receptor 52
Cat. No.: HY-184192
CAS No.: 3066783-67-0
Target:
Research Areas:
R-185 is an orally active and brain-penetrant GPR52 agonist. R-185 activates GPR52 to increase intracellular cAMP levels. R-185 can be used for the research of schizophrenia .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
