1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. nAChR
  3. Zaldaride maleate

Zaldaride maleate (Synonyms: CGS-9343B; KW 5617)

Cat. No.: HY-105118A Purity: >98.0%
Handling Instructions

Zaldaride maleate (CGS-9343B) is a potent and selective inhibitor of calmodulin. Zaldaride maleate (CGS-9343B) inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM. Zaldaride maleate (CGS-9343B) prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR.

For research use only. We do not sell to patients.

Zaldaride maleate Chemical Structure

Zaldaride maleate Chemical Structure

CAS No. : 109826-27-9

Size Price Stock Quantity
10 mM * 1 mL in Water USD 252 In-stock
Estimated Time of Arrival: December 31
5 mg USD 210 In-stock
Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

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Description

Zaldaride maleate (CGS-9343B) is a potent and selective inhibitor of calmodulin. Zaldaride maleate (CGS-9343B) inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM[1][2]. Zaldaride maleate (CGS-9343B) prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR[3].

IC50 & Target

IC50: 3.3 nM (calmodulin)[1][2].

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References
Molecular Weight

544.60

Formula

C₃₀H₃₂N₄O₆

CAS No.

109826-27-9

SMILES

O=C(O)/C=C\C(O)=O.CC1(C2=CC=CN2C3=CC=CC=C3CO1)CN4CCC(N5C6=C(C=CC=C6)NC5=O)CC4

Shipping

Room temperature in continental US; may vary elsewhere

Purity: >98.0%

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Product Name:
Zaldaride maleate
Cat. No.:
HY-105118A
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Zaldaride maleate

Cat. No.: HY-105118A