1. Neuronal Signaling
  2. Serotonin Transporter
  3. Azaphen dihydrochloride monohydrate

Azaphen dihydrochloride monohydrate (Synonyms: Azafen dihydrochloride monohydrate; Pipofezin dihydrochloride monohydrate; Pipofezine dihydrochloride monohydrate; Azaphenonxazine dihydrochloride monohydrate)

Cat. No.: HY-A0022A Purity: 99.60%
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Pipofezine(Azafen or Azaphen) is a potent inhibitor of the reuptake of serotonin.

For research use only. We do not sell to patients.

Azaphen dihydrochloride monohydrate Chemical Structure

Azaphen dihydrochloride monohydrate Chemical Structure

CAS No. : 63302-99-8

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500 mg USD 370 In-stock
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Description

Pipofezine(Azafen or Azaphen) is a potent inhibitor of the reuptake of serotonin. IC50 Value: Target: SSRIs Pipofezine is a tricyclic antidepressant (TCA) approved in Russia for the treatment ofdepression. In addition to its antidepressant action, pipofezine has sedative effects as well, indicating antihistamine activity.

Molecular Weight

388.29

Formula

C₁₆H₂₃Cl₂N₅O₂

CAS No.

63302-99-8

SMILES

[H]Cl.[H]Cl.CN1C2=CC=CC=C2OC3=C1C=C(N4CCN(C)CC4)N=N3.O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

H2O : ≥ 100 mg/mL (257.54 mM)

DMSO : 1 mg/mL (2.58 mM; Need ultrasonic)

*"≥" means soluble, but saturation unknown.

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Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5754 mL 12.8770 mL 25.7539 mL
5 mM 0.5151 mL 2.5754 mL 5.1508 mL
10 mM 0.2575 mL 1.2877 mL 2.5754 mL
*Please refer to the solubility information to select the appropriate solvent.
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The molarity calculator equation

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

Azaphen dihydrochlorideAzafen dihydrochloridePipofezin dihydrochloridePipofezine dihydrochlorideAzaphenonxazine dihydrochlorideSerotonin Transporter5-HTTSERTSLC6A4Inhibitorinhibitorinhibit

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Product Name:
Azaphen dihydrochloride monohydrate
Cat. No.:
HY-A0022A
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