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Edicotinib (Synonyms: JNJ-40346527)

Cat. No.: HY-109086
Handling Instructions

Edicotinib is a selective and orally available colony-stimulating factor-1 (CSF-1) receptor inhibitor, and has entered phase IIA clinical trial to study rheumatoid arthritis (RA) despite disease.

For research use only. We do not sell to patients.

Edicotinib Chemical Structure

Edicotinib Chemical Structure

CAS No. : 1142363-52-7

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  • Biological Activity

  • Technical Information

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  • References

Description

Edicotinib is a selective and orally available colony-stimulating factor-1 (CSF-1) receptor inhibitor, and has entered phase IIA clinical trial to study rheumatoid arthritis (RA) despite disease.

IC50 & Target

CSF-1 receptor[1]

Clinical Trial
Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1664 mL 10.8319 mL 21.6638 mL
5 mM 0.4333 mL 2.1664 mL 4.3328 mL
10 mM 0.2166 mL 1.0832 mL 2.1664 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

461.60

Formula

C₂₇H₃₅N₅O₂

CAS No.

1142363-52-7

SMILES

O=C(C1=NC=C(C#N)N1)NC2=C(C3=CCC(C)(C)CC3)N=C(C(CC(C)(C)O4)CC4(C)C)C=C2

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Edicotinib
Cat. No.:
HY-109086
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Edicotinib

Cat. No.: HY-109086