1. GPCR/G Protein
  2. Oxytocin Receptor
  3. Retosiban

Retosiban (Synonyms: GSK 221149; GSK 221149A)

Cat. No.: HY-14778
Handling Instructions

Retosiban (GSK221149A) is a potent and selective oxytocin antagonist with a Ki of 0.65 nM.

For research use only. We do not sell to patients.

Retosiban Chemical Structure

Retosiban Chemical Structure

CAS No. : 820957-38-8

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Description

Retosiban (GSK221149A) is a potent and selective oxytocin antagonist with a Ki of 0.65 nM.

IC50 & Target

IC50: 0.65 nM (Oxytocin)[1]

Clinical Trial
Molecular Weight

494.58

Formula

C₂₇H₃₄N₄O₅

CAS No.

820957-38-8

SMILES

O=C([[email protected]@H](C1CC2=C(C=CC=C2)C1)N3)N([[email protected]](C4=COC(C)=N4)C(N5CCOCC5)=O)[[email protected]]([[email protected]](CC)C)C3=O

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
Retosiban
Cat. No.:
HY-14778
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