1. GPCR/G Protein
  2. Oxytocin Receptor
  3. Retosiban

Retosiban (Synonyms: GSK 221149; GSK 221149A)

Cat. No.: HY-14778
Handling Instructions

Retosiban (GSK221149A) is a potent and selective oxytocin antagonist with a Ki of 0.65 nM.

For research use only. We do not sell to patients.

Retosiban Chemical Structure

Retosiban Chemical Structure

CAS No. : 820957-38-8

Size Price Stock
5 mg USD 680 Ask For Quote & Lead Time
10 mg USD 1100 Ask For Quote & Lead Time
50 mg USD 3500 Ask For Quote & Lead Time
100 mg USD 5500 Ask For Quote & Lead Time

* Please select Quantity before adding items.

Top Publications Citing Use of Products
  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

Retosiban (GSK221149A) is a potent and selective oxytocin antagonist with a Ki of 0.65 nM.

IC50 & Target

IC50: 0.65 nM (Oxytocin)[1]

Clinical Trial
Molecular Weight

494.58

Formula

C₂₇H₃₄N₄O₅

CAS No.

820957-38-8

SMILES

O=C([[email protected]@H](C1CC2=C(C=CC=C2)C1)N3)N([[email protected]](C4=COC(C)=N4)C(N5CCOCC5)=O)[[email protected]]([[email protected]](CC)C)C3=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • No file chosen (Maximum size is: 1024 Kb)
  • If you have published this work, please enter the PubMed ID.
  • Your name will appear on the site.
  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

RetosibanGSK 221149 GSK 221149AGSK221149GSK-221149Oxytocin ReceptorOXTRInhibitorinhibitorinhibit

Your Recently Viewed Products:

Inquiry Online

Your information is safe with us. * Required Fields.

Product Name

 

Salutation

Applicant Name *

 

Email address *

Phone number *

 

Organization name *

Country or Region *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
Retosiban
Cat. No.:
HY-14778
Quantity:
MCE Japan Authorized Agent: