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Cat. No.: HY-120846

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CHIR 4531

CHIR 4531, a trimer peptide, is a opiate ligand that binds to the mu-opiate receptor with a K_i of 6 nM.

For research use only. We do not sell to patients.

CAS No.: 158198-48-2
Formula: C₃₆H₃₈N₄O₆
Molecular Weight:622.71

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (269 KB)

CHIR 4531 Chemical Structure

CAS No.: 158198-48-2

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

CHIR 4531, a trimer peptide, is a opiate ligand that binds to the mu-opiate receptor with a K_i of 6 nM^[1].

IC₅₀ & Target^[1]

μ Opioid Receptor/MOR

6 nM (Ki)

All Opioid Receptor Isoforms :

Chemical Information

CAS No. 158198-48-2
Molecular Weight 622.71
Formula C₃₆H₃₈N₄O₆
SMILES

O=C(N)CN(C(CN(C(CNCC(C1=CC=CC=C1)C2=CC=CC=C2)=O)CC3=CC=C(OCO4)C4=C3)=O)CCC5=CC=C(O)C=C5
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (269 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. R N Zuckermann, et al. Discovery of nanomolar ligands for 7-transmembrane G-protein-coupled receptors from a diverse N-(substituted)glycine peptoid library. J Med Chem. 1994 Aug 19;37(17):2678-85. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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CHIR 4531

All Opioid Receptor Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

CHIR 4531 Related Classifications

HY-120846 Related Classifications