1. Membrane Transporter/Ion Channel
  2. P2X Receptor
  3. AZ10606120 dihydrochloride

AZ10606120 dihydrochloride 

Cat. No.: HY-108669
Handling Instructions

AZ10606120 dihydrochloride is a selective, high affinity antagonist for P2X7 receptor (P2X7R) at human and rat with an IC50 of ~10 nM. AZ10606120 dihydrochloride is little or no effect at other P2XR subtypes. AZ10606120 dihydrochloride has anti-depressant effects and reduces tumour growth.

For research use only. We do not sell to patients.

AZ10606120 dihydrochloride Chemical Structure

AZ10606120 dihydrochloride Chemical Structure

CAS No. : 607378-18-7

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Description

AZ10606120 dihydrochloride is a selective, high affinity antagonist for P2X7 receptor (P2X7R) at human and rat with an IC50 of ~10 nM. AZ10606120 dihydrochloride is little or no effect at other P2XR subtypes. AZ10606120 dihydrochloride has anti-depressant effects and reduces tumour growth[1].

IC50 & Target

IC50: ~10 nM (P2X7R)[1]

Molecular Weight

495.48

Formula

C₂₅H₃₆Cl₂N₄O₂

CAS No.

607378-18-7

SMILES

O=C(NC1=C2C=CC(NCCNCCO)=NC2=CC=C1)CC3(C4)CC5CC4CC(C5)C3.[H]Cl.[H]Cl

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Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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AZ10606120 dihydrochloride
Cat. No.:
HY-108669
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