Lp(a)-IN-5
Lp(a)-IN-5 (Compound A) is an orally active lipoprotein (a) (Lp(a)) inhibitor. Lp(a)-IN-5 inhibits the assembly of Apo(a) and ApoB proteins with an IC50 value of 0.41 nM. Lp(a)-IN-5 is promising for research of diseases related to elevated plasma Lp(a) levels, such as cardiovascular diseases.
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- CAS No.: 2924841-79-0
- Formule: C43H56N4O7
- Masse moléculaire:740.93
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
| Species | Dose | Route | Cmax | AUC | T1/2 |
|---|---|---|---|---|---|
| Dog[1] | 10 mg/kg | p.o. | 2473 ng/mL | 28594 ng·h/mL | 18.3 h |
Chemical Information
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CAS No. 2924841-79-0
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Masse moléculaire 740.93
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Formule C43H56N4O7
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SMILES
O=C(O)[C@H]([C@H]1CCNC1)CC2=CC=CC(CN(CC3=CC(C[C@H](C(O)=O)[C@H]4CCNC4)=CC=C3)CCOC5=CC(C[C@H](C(O)=O)[C@H]6CCNC6)=CC=C5)=C2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Lp(a)-IN-5 Related Classifications
HY-171464 Related Classifications
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