LSD1/2-IN-4
LSD1/2-IN-4, a PCPA derivative, is an inhibitor of lysine-specific demethylase 1 (LSD1) and lysine-specific demethylase 2 (LSD2). LSD1/2-IN-4 inhibits LSD1 and LSD2 with Ki values of 0.11 μM and 130 μM, respectively. LSD1/2-IN-4 can be used for the research of several cancers including T-cell acute lymphoblastic leukemia (TALL).
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- CAS No.: 2821068-09-9
- Formule: C9H8BrF2N
- Masse moléculaire:248.07
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Help & FAQs
Activité biologique
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KDM1/LSD1 |
LSD1/2-IN-4 shows strong inhibitory activity against both LSD1 and LSD2 with Ki values of 0.11 μM and 130 μM, respectively and not inhibits peroxidase with an IC50 >500 μM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2821068-09-9
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Masse moléculaire 248.07
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Formule C9H8BrF2N
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SMILES
N[C@@H]1C[C@H]1C2=CC(F)=C(Br)C(F)=C2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
LSD1/2-IN-4 Related Classifications
HY-151194 Related Classifications
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