SSTR5 antagonist 2
SSTR5 antagonist 2 (compound 10) is a highly potent, oral active and selective somatostatin (receptor) subtype 5 (SSTR5) antagonist and has potential for the research of treat type 2 diabetes mellitus (T2DM).
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- CAS. Nr.: 1254730-81-8
- Formel: C32H35FN2O5
- Molecular Weight:546.63
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
- Reinheit & Dokumentation
- Verweise
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Help & FAQs
Biologische Aktivität
SSTR5[1].
SSTR5 antagonist 2 increases pancreatic insulin secretion as well as total and active GLP1 release, and demonstrates synergistic effects in combination with DPP4 inhibitors[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Animal Model:Rodent diabetic model without risk of hypoglycemia[1].
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Dosage:10 mg/kg.
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Administration:Orally.
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Result:Increased both total and active circulating incretin hormone GLP1 levels.
Chemical Information
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CAS. Nr. 1254730-81-8
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Molecular Weight 546.63
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Formel C32H35FN2O5
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SMILES
FC(C=C1)=CC=C1C2=C(OCC)C=C(CN3CCC4(CN(C5=CC=C(C(O)=O)C=C5)C(C4)=O)CC3)C=C2OCC
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
SSTR5 antagonist 2 Related Classifications
HY-114191 Related Classifications
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