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Cat. No.: HY-123142

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RX809055AX

RX 809055AX is a potent long lasting opioid antagonist with selectivity towards at mu and delta receptors.

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CAS No.: 122566-12-5
Formule: C₂₉H₂₉ClN₂O₄
Masse moléculaire:505.00

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (275 KB)

RX809055AX Chemical Structure

CAS No.: 122566-12-5

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
- Cellular Effect
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

RX 809055AX is a potent long lasting opioid antagonist with selectivity towards at mu and delta receptors^[1].

IC₅₀ & Target

μ Opioid Receptor/MOR

δ Opioid Receptor/DOR

Voir tous les produits spécifiques à Isoform Opioid Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
CHO	IC₅₀	0.1 nM Compound: 4a, C-CAM	Activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding Activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding	[PMID: 17004724]
CHO	IC₅₀	0.19 nM Compound: 4a, C-CAM	Activity at human recombinant delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding Activity at human recombinant delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding	[PMID: 17004724]
CHO	IC₅₀	0.53 nM Compound: 4a, C-CAM	Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding	[PMID: 17004724]

Chemical Information

CAS No. 122566-12-5
Masse moléculaire 505.00
Formule C₂₉H₂₉ClN₂O₄
SMILES

ClC(C=C1)=CC=C1/C=C/C(N[C@]23[C@@]45C6=C(C[C@@]3([H])N(CC5)CC7CC7)C=CC(O)=C6O[C@@]4([H])C(CC2)=O)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (275 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Lemcke PK, Ayres EA, Kramer TH, Burks TF. RX809055AX in vivo: a long lasting opioid antagonist at mu and delta receptors. Proc West Pharmacol Soc. 1989;32:173-5. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

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MOQ

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100 mg

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Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références

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RX809055AX

Voir tous les produits spécifiques à Isoform Opioid Receptor