KOR agonist 2
KOR agonist 2 (Compound 23p) is an agonist for κ opioid receptor (KOR) with Ki of 1.9 nM. KOR agonist 2 exhibits analgesic effect in mouse models with ED50 of 1.30 mg/kg. KOR agonist 2 exhibits high clearance rate (2 mg/kg, i.v.) in mice, high metabolism and clearance in liver microsomes.
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- No. CAS: 3050912-29-0
- Fòrmula: C29H35ClN2O4S
- Peso molecular:543.12
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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κ Opioid Receptor/KOR 1.9 nM (Ki) |
Chemical Information
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No. CAS 3050912-29-0
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Peso molecular 543.12
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Fòrmula C29H35ClN2O4S
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SMILES
O=S(C1=CC=CC(Cl)=C1)(N(CC2=CC=CC=C2)[C@@H]3C[C@H](CN(C)C)[C@](C4=CC=CC(OC)=C4)(O)CC3)=O
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
KOR agonist 2 Related Classifications
HY-159088 Related Classifications
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